ETINACT-P
Composition: Etoricoxib 60mg+Paracetamol 325mg
Indication: Arthritis , Post Surgical Pain Management, Spondylitis, Acute Low Back Pain.
Packing: 10x10
Pack Type: Tab

Description

ETINACT-P TABS (Etoricoxib Paracetamol) – Comprehensive Overview

Introduction

ETINACT-P TABS is a powerful combination medication containing Etoricoxib Paracetamol. This formulation is widely used for pain relief, inflammation reduction, and fever control. It is commonly prescribed for conditions like arthritis, musculoskeletal pain, and post-operative discomfort. Etoricoxib is a selective COX-2 inhibitor that provides anti-inflammatory and analgesic effects, while Paracetamol works as an antipyretic and mild analgesic, enhancing the overall effectiveness of the medication.

Composition

Each ETINACT-P TAB contains:

  • Etoricoxib – A selective COX-2 inhibitor that helps reduce inflammation and pain.
  • Paracetamol – A widely used analgesic and antipyretic agent that enhances pain relief and fever control.

Mechanism of Action

  • Etoricoxib: This molecule selectively inhibits the cyclooxygenase-2 (COX-2) enzyme, reducing prostaglandin synthesis. This action helps in alleviating pain and inflammation without significantly affecting COX-1, which maintains gastrointestinal protection.
  • Paracetamol: Works by inhibiting prostaglandin synthesis in the central nervous system, providing pain relief and fever reduction. It complements Etoricoxib, ensuring enhanced efficacy with a balanced safety profile.

Indications

ETINACT-P TABS is recommended for various painful and inflammatory conditions, including:

  • Osteoarthritis – Provides symptomatic relief from joint pain and stiffness.
  • Rheumatoid Arthritis – Helps in reducing chronic inflammation and pain.
  • Ankylosing Spondylitis – Alleviates spinal pain and stiffness.
  • Post-operative Pain – Used for acute pain management after surgery.
  • Musculoskeletal Disorders – Effective in treating conditions like sprains, strains, and tendonitis.
  • Dental Pain – Reduces post-extraction or post-surgical dental discomfort.
  • Fever and Mild-to-Moderate Pain – Helps in managing fever and general body pain.

Dosage and Administration

  • The recommended dosage of ETINACT-P TABS depends on the severity of the condition and medical advice.
  • It should be taken with food or water to reduce gastric irritation.
  • Etoricoxib Paracetamol combination should not exceed the prescribed dosage to avoid potential side effects.

Benefits of ETINACT-P TABS

  • Dual Action: Provides effective pain relief by combining Etoricoxib and Paracetamol.
  • Reduced Gastrointestinal Effects: Unlike traditional NSAIDs, Etoricoxib selectively inhibits COX-2, minimizing the risk of gastric ulcers.
  • Enhanced Pain Management: The combination of Etoricoxib Paracetamol ensures comprehensive pain relief.
  • Faster Onset of Action: Provides quick relief from pain and fever.
  • Convenient Dosing: Single tablet formulation improves patient compliance.

Side Effects

While generally well-tolerated, some patients may experience:

  • Gastrointestinal Issues – Nausea, vomiting, dyspepsia, or gastric irritation.
  • Cardiovascular Risks – Long-term use of Etoricoxib may slightly increase the risk of heart-related issues.
  • Liver ConcernsParacetamol in high doses can lead to hepatotoxicity.
  • Allergic Reactions – Skin rashes, itching, or swelling in rare cases.

Precautions & Warnings

  • Not Recommended in Patients with Peptic Ulcers: Etoricoxib Paracetamol should be used cautiously in individuals with a history of gastric ulcers or bleeding disorders.
  • Use in Hepatic or Renal Impairment: Dose adjustments may be required for patients with liver or kidney dysfunction.
  • Pregnancy & Lactation: Consult a healthcare professional before use during pregnancy or breastfeeding.
  • Avoid Alcohol Consumption: Alcohol can enhance liver toxicity risks when combined with Paracetamol.
  • Caution in Cardiovascular Patients: Prolonged use should be monitored due to possible heart risks.

Drug Interactions

  • Antihypertensives: Etoricoxib may reduce the effectiveness of blood pressure medications.
  • Anticoagulants: Increased risk of bleeding when combined with warfarin or similar drugs.
  • Other NSAIDs: Avoid concurrent use to prevent excessive gastric irritation.
  • Liver Enzyme Inducers: Drugs like rifampicin may alter Etoricoxib Paracetamol metabolism.

Conclusion

ETINACT-P TABS is a clinically effective pain-relief medication combining Etoricoxib Paracetamol to provide dual-action relief from pain, inflammation, and fever. With its selective COX-2 inhibition and added Paracetamol benefits, it is a preferred choice for managing arthritis, musculoskeletal disorders, post-operative pain, and general fever management. Proper usage as per medical guidance ensures maximum efficacy with minimal side effects.

Disclaimer: This content is for informational purposes only. Consult your healthcare provider before using ETINACT-P TABS or any medication containing Etoricoxib Paracetamol.

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